{"id":995,"date":"2020-12-03T10:49:19","date_gmt":"2020-12-03T01:49:19","guid":{"rendered":"https:\/\/www.promega.co.jp\/resources\/faq\/?p=995"},"modified":"2021-01-20T13:08:18","modified_gmt":"2021-01-20T04:08:18","slug":"q747","status":"publish","type":"post","link":"https:\/\/www.promega.co.jp\/resources\/faq\/cell-health\/adme\/p450\/p450-glo\/q747","title":{"rendered":"CYP450\u306e\u963b\u5bb3\u5264\u3068\u3057\u3066\u77e5\u3089\u308c\u3066\u3044\u308b\u5316\u5408\u7269\u3092\u4f7f\u7528\u3057\u305f\u5834\u5408\u306b\u3082\u304b\u304b\u308f\u3089\u305a\u3001CYP450\u306e\u53cd\u5fdc\u304c\u963b\u5bb3\u3055\u308c\u306a\u304b\u3063\u305f\u4e8b\u4f8b\u306f\u3042\u308a\u307e\u3059\u304b\uff1f"},"content":{"rendered":"\n<p>CYP3A4 \u963b\u5bb3\u5264\u306eTerfenadine(\u6297\u30a2\u30ec\u30eb\u30ae\u30fc\u85ac) \u3092\u6dfb\u52a0\u3057\u305f\u3068\u304d\u306b\u3001\u7cbe\u88fd\u9175\u7d20\u306e\u307f\u3068\u6bd4\u8f03\u3057\u3066\u3001RLU\u5024\u304c2\u500d\u4e0a\u6607\u3057\u305f\u3053\u3068\u304c\u5831\u544a\u3055\u308c\u3066\u3044\u307e\u3059\u3002CYP3A4\u306b\u306f\u3001\u9175\u7d20\u89e6\u5a92\u306e\u6d3b\u6027\u90e8\u4f4d\u304c\u591a\u6570\u3042\u308b\u305f\u3081\u3001\u3053\u306e\u5834\u5408\u306f\u3001Terfenadine\u5358\u72ec\u3067\u306fCYP3A4\u306e\u6d3b\u6027\u3092\u963b\u5bb3\u3067\u304d\u306a\u304b\u3063\u305f\u305f\u3081\u3060\u3068\u8003\u3048\u3089\u308c\u3066\u3044\u307e\u3059\u3002\u305f\u3060\u3057\u3001\u7cbe\u88fd\u9175\u7d20\u3092\u5358\u72ec\u4f7f\u7528\u3057\u305f\u3068\u304d\u3068\u6bd4\u3079\u3066\u3001RLU\u5024\u304c\u4e0a\u6607\u3057\u305f\u3053\u3068\u306b\u3064\u3044\u3066\u306e\u539f\u56e0\u306f\u4e0d\u660e\u3067\u3059\u3002<\/p>\n\n\n\n<p>CYP450\u306e\u53cd\u5fdc\u963b\u5bb3\u306f\u3001 \u751f\u4f53\u5185\u306e\u4ee3\u8b1d\u3084\u8907\u6570\u306e\u57fa\u8cea\u304c\u5b58\u5728\u3059\u308b\u3053\u3068\u306b\u3088\u308a\u3001\u751f\u3058\u308b\u3068\u3055\u308c\u3066\u3044\u307e\u3059\u3002\u963b\u5bb3\u5264\u306e\u30b9\u30af\u30ea\u30fc\u30cb\u30f3\u30b0\u6642\u306b\u3001\u671f\u5f85\u306b\u53cd\u3057\u305f\u7d50\u679c\u304c\u8a8d\u3081\u3089\u308c\u305f\u5834\u5408\u306f\u3001\u8907\u6570\u306e\u7570\u306a\u308b\u57fa\u8cea\u306e\u4f7f\u7528\u3084\u3001P450-Glo\u2122 Assay\u4ee5\u5916\u306e\u6e2c\u5b9a\u65b9\u6cd5\uff08\u86cd\u5149\u6cd5\u306a\u3069\uff09\u3092\u5b9f\u65bd\u3057\u3001\u7dcf\u5408\u7684\u306b\u8a55\u4fa1\u3059\u308b\u3053\u3068\u3092\u304a\u85a6\u3081\u3044\u305f\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<p>\u306a\u304a\u3001\u73fe\u5728\u8ca9\u58f2\u3055\u308c\u3066\u3044\u308bP450-Glo\u2122 Assay\u306e\u5404CYP450\u5206\u5b50\u7a2e\u306b\u5bfe\u3059\u308b\u963b\u5bb3\u5264\uff08\u5316\u5408\u7269\uff09\u306e\u30ea\u30b9\u30c8\u304c\u3042\u308a\u307e\u3059\uff081\uff09\u3002<\/p>\n\n\n\n<p>\u53c2\u8003\u6587\u732e<br>1. Cali, J.S. et al. (2006) Luminogenic cytochrome P450 assays. Expert. Opin. Drug. Metab. Toxicol. 2, 629-45.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>CYP3A4 \u963b\u5bb3\u5264\u306eTerfenadine(\u6297\u30a2\u30ec\u30eb\u30ae\u30fc\u85ac) \u3092\u6dfb\u52a0\u3057\u305f\u3068\u304d\u306b\u3001\u7cbe\u88fd\u9175\u7d20\u306e\u307f\u3068\u6bd4\u8f03\u3057\u3066\u3001RLU\u5024\u304c2\u500d\u4e0a\u6607\u3057\u305f\u3053\u3068\u304c\u5831\u544a\u3055\u308c\u3066\u3044\u307e\u3059\u3002CYP3A4\u306b\u306f\u3001\u9175\u7d20\u89e6\u5a92\u306e\u6d3b\u6027\u90e8\u4f4d\u304c\u591a\u6570\u3042\u308b\u305f\u3081\u3001\u3053\u306e\u5834\u5408\u306f\u3001Te &#8230; <\/p>\n","protected":false},"author":16,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":[],"categories":[235],"tags":[],"_links":{"self":[{"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/posts\/995"}],"collection":[{"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/users\/16"}],"replies":[{"embeddable":true,"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/comments?post=995"}],"version-history":[{"count":1,"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/posts\/995\/revisions"}],"predecessor-version":[{"id":996,"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/posts\/995\/revisions\/996"}],"wp:attachment":[{"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/media?parent=995"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/categories?post=995"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/www.promega.co.jp\/resources\/faq\/wp-json\/wp\/v2\/tags?post=995"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}